SARMs selective androgen receptor modulators
Selective androgen receptor modulators or SARMs are a novel class of androgen receptor ligands. (The name follows the terminology currently used for similar molecules targeting the estrogen receptor, "selective estrogen receptor modulators," such as Tamoxifen.) They are intended to have the same kind of effects as androgenic drugs like anabolic steroids but be much more selective in their action, allowing them to be used for many more clinical indications than the relatively limited legitimate uses that anabolic steroids are currently approved for.
Currently used androgens for male hormone replacement therapy are typically injectable or skin delivery formulations of testosterone or testosterone esters. Injectable forms of testosterone esters (such as testosterone enanthate, propionate, or cypionate) produce undesirable fluctuations in testosterone blood levels, with overly high levels shortly after injection and overly low afterward. Skin patches do provide a better blood level profile of testosterone, but skin irritation and daily application still limit their usefulness.
SARMs provide the opportunity to design molecules that can be delivered orally, but that selectively target the androgen receptors in different tissues differently. The goal of research in this area is to allow a customized response: Tissues that are the target of the therapy will respond as they would to testosterone; other tissues where undesirable side-effects are produced will not.
Selective Androgen Receptor Modulators : Every Bodybuilders Wet Dream Come True SARMS have full anabolic activity in muscle and bone, yet have minimal effect the on prostate. SARMS are highly specific to the androgen receptor as they have a 1000-fold less binding affinity for any other receptor
Ockham’s Razor and Selective Androgen Receptor Modulators (SARMs): Are We Overlooking the Role of 5a-Reductase considerable progress in the discovery and development of SARMs in the past decade with SARMs having much improved specificity for androgen receptor
Expanding the therapeutic use of androgens via selective androgen receptor modulators (SARMs) Research into SARMs has made dramatic progress over the past decade efforts continue to be devoted to nonsteroidal AR agonists as anabolic SARMs
Selective Androgen Receptor Modulators (SARMs) Promoting Anabolic Therapies SARMs hold considerable promise as a new class of function promoting anabolic therapies through the Mechanisms of SARM Tissue Selectivity
Bodybuilding Muscle Mass SARM LGD-4033 LGD-4033 is an oral SARM that is non-steroidal, but it can offer many of the same benefits as some of the anabolic steroids. The use of LGD-4033 medically includes treatment of muscle wasting.
Anabolic bodybuilding muscle mass SARM Andarine S4 This anabolic bodybuilding musle mass SARM can help with creating lean body mass. Andarine S4 can also help with increasing the amount of lean muscle mass
Bodybuilding SARM Enobosarm Ostarine MK-2866 Ostarine is one of the most favorable of any bodybuilding SARMS for being the most anabolic. Of course you can not campare it to anabolic steroids. But in one aspect, you also see none of the side effects you would see with steroids
Ostarine MK-2866 A type of SARM,short for Selective Androgen Receptor Modulator, is called Ostarine MK – 2866. It is typically prescribed for the treatment and prevention of muscle wasting
Anti-Estrogens used as a fat burning cycle Most people have heard of Anti-E's due to their role in a person's steroid cycle. Anti-Estrogens are used to prevent gynocomastia from steroids that aromatize and also reduce water retention. However, Anti-Estrogens can be also used for a host of other reasons, and in our case, fat loss
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